List of combined sex-hormonal preparations
This is a list of known combined sex-hormonal formulations. Brand names and developmental code names are in parentheses.
Androgens
Injection
Marketed
- Nandrolone decanoate/nandrolone phenylpropionate
- Testosterone propionate/testosterone isocaproate/testosterone caproate
- Testosterone propionate/testosterone enanthate/testosterone undecylenate
- Testosterone propionate/testosterone enanthate
- Testosterone propionate/testosterone ketolaurate
- Testosterone propionate/testosterone phenylpropionate/testosterone isocaproate
- Testosterone propionate/testosterone phenylpropionate/testosterone isocaproate/testosterone caproate
- Testosterone propionate/testosterone phenylpropionate/testosterone isocaproate/testosterone decanoate
- Testosterone propionate/testosterone valerate/testosterone undecylenate
- Testosterone propionate/testosterone cypionate/prasterone
Veterinary
Marketed
- Boldenone acetate/boldenone cypionate/boldenone propionate/boldenone undecylenate
- Testosterone acetate/testosterone undecanoate/testosterone valerate
Estrogens
Oral
Marketed
- Conjugated estriol
- Conjugated estrogens
- Esterified estrogens
- Estradiol/estrone/estriol
- Ethinylestradiol/dienestrol
Injection
Marketed
- Estradiol benzoate/estradiol phenylpropionate
Never marketed
- Estradiol/estradiol enanthate
Progestogens
Injection
Marketed
- Progesterone/hydroxyprogesterone heptanoate/α-tocopherol palmitate
Androgens and estrogens
Oral
Marketed
- Chlorotrianisene/methyltestosterone
- Conjugated estrogens/methyltestosterone
- Dienestrol/methyltestosterone
- Dienestrol diacetate/methyltestosterone
- Diethylstilbestrol/methyltestosterone
- Esterified estrogens/methyltestosterone
- Ethinylestradiol/methyltestosterone
- Methylestradiol/methyltestosterone
- Methylestradiol/methyltestosterone/reserpine
Injection
Marketed
- Estradiol benzoate/testosterone propionate
- Estradiol benzoate/estradiol dienanthate/testosterone enanthate benzilic acid hydrazone
- Estradiol benzoate/estradiol phenylpropionate/testosterone propionate/testosterone phenylpropionate/testosterone isocaproate
- Estradiol benzoate/testosterone isobutyrate
- Estradiol butyrylacetate/testosterone ketolaurate/reserpine
- Estradiol cypionate/testosterone cypionate
- Estradiol cypionate/testosterone enanthate
- Estradiol valerate/prasterone enanthate
- Estradiol valerate/testosterone enanthate
Veterinary
Marketed
- Diethylstilbestrol/methyltestosterone
- Diethylstilbestrol/testosterone
- Estradiol benzoate/estradiol enanthate/testosterone enanthate
- Estradiol benzoate/testosterone propionate
- Ethinylestradiol/methyltestosterone
Estrogens and progestogens
Oral
Marketed
In birth control pills:- Estradiol/nomegestrol acetate
- Estradiol valerate/cyproterone acetate
- Estradiol valerate/dienogest
- Ethinylestradiol/chlormadinone acetate
- Ethinylestradiol/cyproterone acetate
- Ethinylestradiol/desogestrel
- Ethinylestradiol/dienogest
- Ethinylestradiol/dimethisterone
- Ethinylestradiol/drospirenone
- Ethinylestradiol/drospirenone/levomefolic acid
- Ethinylestradiol/etynodiol diacetate
- Ethinylestradiol/gestodene
- Ethinylestradiol/levonorgestrel
- Ethinylestradiol/levonorgestrel/bisglycinate
- Ethinylestradiol/levonorgestrel/ferrous fumarate
- Ethinylestradiol/lynestrenol
- Ethinylestradiol/medroxyprogesterone acetate
- Ethinylestradiol/megestrol acetate
- Ethinylestradiol/norethisterone
- Ethinylestradiol/norethisterone/ferrous fumarate
- Ethinylestradiol/norethisterone acetate
- Ethinylestradiol/norethisterone acetate/ferrous fumarate
- Ethinylestradiol/norgestimate
- Ethinylestradiol/norgestrel
- Ethinylestradiol/norgestrienone
- Ethinylestradiol/quingestanol acetate
- Ethinylestradiol sulfonate/norethisterone acetate
- Mestranol/anagestone acetate
- Mestranol/chlormadinone acetate
- Mestranol/etynodiol diacetate
- Mestranol/hydroxyprogesterone acetate
- Mestranol/lynestrenol
- Mestranol/norethisterone
- Mestranol/noretynodrel
- Quinestrol/etynodiol diacetate
- Quinestrol/levonorgestrel
- Quinestrol/norgestrel
- Quinestrol/quingestanol acetate
- Conjugated estrogens/medrogestone
- Conjugated estrogens/medroxyprogesterone acetate
- Conjugated estrogens/norgestrel
- Estradiol/drospirenone
- Estradiol/dydrogesterone
- Estradiol/gestodene
- Estradiol/levonorgestrel
- Estradiol/medroxyprogesterone acetate
- Estradiol/norethisterone acetate
- Estradiol/norgestimate
- Estradiol/progesterone
- Estradiol/trimegestone
- Estradiol valerate/cyproterone acetate
- Estradiol valerate/estriol/levonorgestrel
- Estradiol valerate/levonorgestrel
- Estradiol valerate/medroxyprogesterone acetate
- Estradiol valerate/norethisterone
- Estradiol valerate/norethisterone acetate
- Estradiol valerate/norgestrel
- Ethinylestradiol/ethisterone
- Mestranol/noretynodrel
Never or not yet marketed
- Estetrol/drospirenone
- Estradiol/norethisterone
Transdermal
Marketed
In contraceptive patches:For menopausal hormone therapy:
- Estradiol/levonorgestrel
- Estradiol/norethisterone acetate
Vaginal
Marketed
In contraceptive vaginal rings:Marketed
In combined injectable contraceptives:- Estradiol/megestrol acetate
- Estradiol benzoate/estradiol valerate/hydroxyprogesterone caproate
- Estradiol benzoate butyrate/algestone acetophenide
- Estradiol cypionate/hydroxyprogesterone caproate
- Estradiol cypionate/medroxyprogesterone acetate
- Estradiol enanthate/algestone acetophenide
- Estradiol valerate/hydroxyprogesterone caproate
- Estradiol valerate/norethisterone enanthate
- Estradiol/progesterone
- Estradiol benzoate/hydroxyprogesterone caproate
- Estradiol benzoate/progesterone
- Estradiol dipropionate/hydroxyprogesterone caproate
- Estradiol hemisuccinate/progesterone
- Estradiol pivalate/progesterone
- Estradiol valerate/hydroxyprogesterone caproate
- Estrone/progesterone
Never marketed
- Estradiol undecylate/norethisterone enanthate
- Estradiol valerate/methenmadinone caproate
- Polyestradiol phosphate/medroxyprogesterone acetate
- Additional preparations listed at Combined injectable birth control § Research
- Estradiol valerate/gestonorone caproate
Veterinary
Marketed
- Estradiol benzoate/progesterone
- Estradiol valerate/norgestomet
Androgens and progestogens
Oral
Marketed
- Methyltestosterone/ethisterone
Injection
Marketed
- Testosterone propionate/progesterone
Veterinary
Marketed
- Danazol/megestrol acetate
- Nandrolone decanoate/methandriol dipropionate
- Nandrolone phenylpropionate/methandriol dipropionate
Estrogens, progestogens, and androgens
Oral
Marketed
- Methylestradiol/normethandrone
Not yet marketed
- Ethinylestradiol/drospirenone/prasterone
Sublingual
Marketed
Marketed
- Estradiol benzoate/progesterone/methandriol dipropionate
- Estradiol benzoate/progesterone/testosterone propionate
- Estradiol benzoate/estradiol valerate/norethisterone acetate/testosterone enanthate
- Estradiol dibutyrate/hydroxyprogesterone heptanoate/testosterone caproate
- Estradiol diundecylate/hydroxyprogesterone heptanoate/testosterone cyclohexylpropionate
- Estradiol hexahydrobenzoate/hydroxyprogesterone caproate/testosterone hexahydrobenzoate
- Estrone/progesterone/testosterone
Never marketed
- Estrapronicate/hydroxyprogesterone heptanoate/nandrolone undecanoate
Veterinary